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Search Results for " h3 receptor antagonist 1 "

9

Compounds

Cat No. Product Name Synonyms Targets
T10911 H3 receptor antagonist 1 Histamine Receptor
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
T79500 KSK94 Histamine Receptor
KSK94 is a specific H3 receptor antagonist that inhibits H3, sigma-1, and sigma-2 receptors , with Ki values of 7.9, 2958, and 75.2 nM, respectively, and can be used to study injurious pain and neuropathic pain.
T79499 KSK68 Histamine Receptor
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 receptors.KSK68 can be used in the study of pain related diseases...
T14087 ABT-239 TRP/TRPV Channel
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists. It also acts as a transient receptor potential vanilloid type 1 (TRPV1) antagonist.
T26643 Aplysamine-1 Aplysamine
Aplysamine-1 is an antagonist of histamine H3 receptor.
T60340 ROS 234
ROS 234 is a highly effective H3 antagonist, demonstrating a strong binding affinity (pK B) of 9.46 for the Guinea-pig ileum H3 receptor and a pKi of 8.90 for the Rat cerebral cortex H3 receptor. Additionally, it exhibit...
T78734 Sigma-1 receptor antagonist 5 Sigma receptor
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptors (Ki=4.5 nM (σ1R), 10 nM (σ2R)) and the histamine H3 receptor...
T61603 H3R antagonist 2
H3R antagonist 2 (Compound 23) is a multitarget histamine H3 receptor antagonist. It exhibits inhibitory effects on acetylcholinesterase, butyrylcholinesterase, and human monoamine oxidase B (hMAO B) with IC50 values of ...
T10462L Bavisant dihydrochloride hydrate JNJ31001074AAC Others
Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wakefulness and cognition, with potential as a treatm...
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